{"id":432,"date":"2026-05-08T14:51:43","date_gmt":"2026-05-08T12:51:43","guid":{"rendered":"https:\/\/doktorpeptid.sk\/?post_type=product&#038;p=432"},"modified":"2026-09-24T14:26:38","modified_gmt":"2026-09-24T12:26:38","slug":"tesamorelin","status":"publish","type":"product","link":"https:\/\/doktorpeptid.sk\/en\/product\/tesamorelin\/","title":{"rendered":"Tesamorelin (TH9507) \u2013 v\u00fdskumn\u00fd peptid 5 mg a 10 mg"},"content":{"rendered":"<h2>Tesamorelin (TH9507) \u2013 v\u00fdskumn\u00fd peptid skladom na Slovensku<\/h2>\n<p><strong>Tesamorelin<\/strong> je syntetick\u00fd anal\u00f3g horm\u00f3nu uvo\u013e\u0148uj\u00faceho rastov\u00fd horm\u00f3n (GHRH), v odbornej literat\u00fare veden\u00fd aj pod k\u00f3dov\u00fdm ozna\u010den\u00edm <strong>TH9507<\/strong>. Ide o 44-aminokyselinov\u00fd re\u0165azec so stabilizuj\u00facou trans-3-hexenoylovou skupinou na N-konci, v\u010faka ktorej je molekula v roztoku odolnej\u0161ia vo\u010di enzymatick\u00e9mu \u0161tiepeniu ne\u017e prirodzen\u00fd GHRH(1\u201344). Pr\u00e1ve t\u00e1to \u00faprava je d\u00f4vodom, pre\u010do sa Tesamorelin objavuje v experiment\u00e1lnych modeloch ako referen\u010dn\u00e1 l\u00e1tka pri \u0161t\u00fadiu osi GHRH \u2013 hypof\u00fdza \u2013 IGF-1.<\/p>\n<p>Dod\u00e1vame ho <strong>lyofilizovan\u00fd<\/strong> v sklenenej ampulke so silik\u00f3novou z\u00e1tkou a hlin\u00edkov\u00fdm uz\u00e1verom, v dvoch ve\u013ekostiach balenia: <strong>5 mg (35,00 \u20ac)<\/strong> a <strong>10 mg (65,00 \u20ac)<\/strong>.<\/p>\n<h2>Mechanizmus, ktor\u00fd sa v literat\u00fare sk\u00fama<\/h2>\n<p>Tesamorelin sa v publikovan\u00fdch modeloch via\u017ee na GHRH receptory v prednom laloku hypof\u00fdzy. Naviazanie sp\u00fa\u0161\u0165a kask\u00e1du cez cyklick\u00fd AMP a vedie k pulzn\u00e9mu uvo\u013e\u0148ovaniu endog\u00e9nneho rastov\u00e9ho horm\u00f3nu. Na rozdiel od priameho podania rastov\u00e9ho horm\u00f3nu zost\u00e1va pri tomto mechanizme zachovan\u00e1 prirodzen\u00e1 pulzatilita sekr\u00e9cie aj sp\u00e4tnov\u00e4zbov\u00e1 regul\u00e1cia cez somatostat\u00edn \u2013 a pr\u00e1ve t\u00e1to vlastnos\u0165 je d\u00f4vodom, pre\u010do je l\u00e1tka v experiment\u00e1lnej endokrinol\u00f3gii sledovan\u00e1.<\/p>\n<p>Sekund\u00e1rne sa v \u0161t\u00fadi\u00e1ch sleduje vplyv na hladiny IGF-1 a na distrib\u00faciu viscer\u00e1lneho tukov\u00e9ho tkaniva. V\u00fdsledky s\u00fa predmetom prebiehaj\u00faceho v\u00fdskumu a nepredstavuj\u00fa tvrdenie o \u00fa\u010dinku u \u013eud\u00ed.<\/p>\n<h2>\u0160pecifik\u00e1cia produktu<\/h2>\n<table>\n<tr>\n<th>N\u00e1zov<\/th>\n<td>Tesamorelin (TH9507)<\/td>\n<\/tr>\n<tr>\n<th>CAS<\/th>\n<td>218949-48-5<\/td>\n<\/tr>\n<tr>\n<th>Sum\u00e1rny vzorec<\/th>\n<td>C221H366N72O67S<\/td>\n<\/tr>\n<tr>\n<th>Mol\u00e1rna hmotnos\u0165<\/th>\n<td>\u2248 5 135,9 g\/mol<\/td>\n<\/tr>\n<tr>\n<th><\/th>\n<td>\u2265 99 %<\/td>\n<\/tr>\n<tr>\n<th>Forma<\/th>\n<td>lyofilizovan\u00fd biely pr\u00e1\u0161ok<\/td>\n<\/tr>\n<tr>\n<th>Balenie<\/th>\n<td>5 mg \/ 10 mg v ampulke<\/td>\n<\/tr>\n<tr>\n<th>Ur\u010denie<\/th>\n<td>v\u00fdhradne laborat\u00f3rny a analytick\u00fd v\u00fdskum<\/td>\n<\/tr>\n<\/table>\n<h2>Rekon\u0161tit\u00facia a manipul\u00e1cia v laborat\u00f3riu<\/h2>\n<p>Lyofiliz\u00e1t sa \u0161tandardne rozp\u00fa\u0161\u0165a <a href=\"\/en\/product\/bakterio-staticka-voda\/\">bakteriostatickou vodou<\/a> (0,9 % benzylalkohol), pr\u00edpadne sterilnou vodou na injekciu, ak sa roztok spotrebuje naraz. Rozp\u00fa\u0161\u0165adlo sa prid\u00e1va pomaly po vn\u00fatornej stene ampulky \u2013 nie priamo na pr\u00e1\u0161ok. Ampulkou sa <strong>nikdy netrepe<\/strong>; peptidov\u00fd re\u0165azec je citliv\u00fd na mechanick\u00e9 nam\u00e1hanie a penenie. Nechajte ju st\u00e1\u0165 pri izbovej teplote, k\u00fdm sa obsah samovo\u013ene nerozpust\u00ed, a potom ju jemne ot\u00e1\u010dajte medzi prstami.<\/p>\n<p>Pri pr\u00e1ci pou\u017e\u00edvajte nesteriln\u00e9 rukavice a\u017e po steriln\u00fa techniku pod\u013ea intern\u00e9ho protokolu v\u00e1\u0161ho pracoviska. Z\u00e1tku pred ka\u017ed\u00fdm odberom dezinfikujte izopropylalkoholom a nechajte oschn\u00fa\u0165.<\/p>\n<h2>Skladovanie a stabilita<\/h2>\n<ul>\n<li><strong>Nerozpusten\u00fd lyofiliz\u00e1t:<\/strong> \u221220 \u00b0C, chr\u00e1nen\u00fd pred svetlom a vlhkos\u0165ou. V tomto stave je peptid stabiln\u00fd dlhodobo.<\/li>\n<li><strong>Kr\u00e1tkodobo pri transporte:<\/strong> izbov\u00e1 teplota po dobu nieko\u013ek\u00fdch dn\u00ed.<\/li>\n<li><strong>Po rekon\u0161tit\u00facii:<\/strong> 2 \u2013 8 \u00b0C v chladni\u010dke, chr\u00e1nen\u00e9 pred svetlom. Roztok nezmrazujte a nevystavujte opakovan\u00fdm cyklom zmrazenia a rozmrazenia.<\/li>\n<\/ul>\n<h2>Balenie a doru\u010denie<\/h2>\n<p>Produkt posielame v pevnom balen\u00ed zabezpe\u010denom proti po\u0161kodeniu po\u010das prepravy.<\/p>\n<p>Certifik\u00e1ty anal\u00fdzy (COA) k jednotliv\u00fdm \u0161ar\u017eiam n\u00e1jdete v sekcii <a href=\"\/en\/coa\/\">Dokumenty COA<\/a>.<\/p>\n<h2>Tesamorelin vs. Ipamorelin \u2013 rozdiel vo v\u00fdskume<\/h2>\n<p>Obe l\u00e1tky sa sk\u00famaj\u00fa v s\u00favislosti s osou rastov\u00e9ho horm\u00f3nu, no p\u00f4sobia cez odli\u0161n\u00e9 receptory. <strong>Tesamorelin<\/strong> je anal\u00f3g GHRH a via\u017ee sa na receptor GHRH (GHRH-R) v prednom laloku hypof\u00fdzy. <a href=\"\/en\/product\/ipamorelin\/\">Ipamorelin<\/a> je pentapeptid zo skupiny sekretag\u00f3gov rastov\u00e9ho horm\u00f3nu (GHRP) a p\u00f4sob\u00ed cez receptor ghrel\u00ednu (GHS-R1a). Preto sa v experiment\u00e1lnych modeloch \u010dasto porovn\u00e1vaj\u00fa alebo sk\u00famaj\u00fa spolo\u010dne. \u010eal\u0161ie l\u00e1tky n\u00e1jdete v kateg\u00f3rii <a href=\"\/en\/product-category\/rastove-peptidy\/\">rastov\u00e9 peptidy<\/a>.<\/p>\n<h2>Tesamorelin peptid na Slovensku a v \u010cesku<\/h2>\n<p>Tesamorelin m\u00e1me <strong>skladom na Slovensku<\/strong> \u2013 objedn\u00e1vku neposielame zo zahrani\u010dn\u00e9ho skladu, ale expedujeme ju spravidla do 24 hod\u00edn. Doru\u010dujeme po celom Slovensku, do \u010ceskej republiky aj do \u010fal\u0161\u00edch kraj\u00edn E\u00da. Na rekon\u0161tit\u00faciu v laborat\u00f3riu odpor\u00fa\u010dame <a href=\"\/en\/product\/bakterio-staticka-voda\/\">bakteriostatick\u00fa vodu 10 ml<\/a>. Ak s peptidmi len za\u010d\u00ednate, pozrite si n\u00e1\u0161ho <a href=\"\/en\/peptidy\/\">sprievodcu peptidmi<\/a>.<\/p>\n<h2>Doprava, platba a vr\u00e1tenie<\/h2>\n<p>Objedn\u00e1vky prijat\u00e9 v pracovn\u00fd de\u0148 odosielame <strong>do 24 hod\u00edn<\/strong>. Doprava na Slovensku od 3,30 \u20ac, pri objedn\u00e1vke nad 150 \u20ac zadarmo. Platba kartou alebo prevodom. Tovar m\u00f4\u017eete vr\u00e1ti\u0165 do 14 dn\u00ed od doru\u010denia.<\/p>\n<h2>Frequently asked questions<\/h2>\n<h3>\u010co je Tesamorelin?<\/h3>\n<p>Tesamorelin (TH9507) je syntetick\u00fd 44-aminokyselinov\u00fd anal\u00f3g GHRH so stabilizuj\u00facou trans-3-hexenoylovou skupinou. V na\u0161ej ponuke je ako lyofilizovan\u00fd peptid ur\u010den\u00fd v\u00fdhradne na laborat\u00f3rny v\u00fdskum.<\/p>\n<h3>Ako Tesamorelin funguje v sk\u00faman\u00fdch modeloch?<\/h3>\n<p>Via\u017ee sa na GHRH receptory hypof\u00fdzy a v publikovan\u00fdch modeloch stimuluje pulzn\u00e9 uvo\u013e\u0148ovanie endog\u00e9nneho rastov\u00e9ho horm\u00f3nu pri zachovan\u00ed prirodzenej sp\u00e4tnej v\u00e4zby.<\/p>\n<h3>V ak\u00fdch ve\u013ekostiach balenia Tesamorelin dod\u00e1vate?<\/h3>\n<p>V dvoch: 5 mg za 35,00 \u20ac a 10 mg za 65,00 \u20ac. Obe s\u00fa skladom na Slovensku.<\/p>\n<h3>\u010c\u00edm sa Tesamorelin rekon\u0161tituuje?<\/h3>\n<p>Naj\u010dastej\u0161ie bakteriostatickou vodou s 0,9 % benzylalkoholu. Rozp\u00fa\u0161\u0165adlo sa prid\u00e1va po stene ampulky, obsahom sa netrepe.<\/p>\n<h3>Ako sa Tesamorelin skladuje?<\/h3>\n<p>Lyofiliz\u00e1t pri \u221220 \u00b0C chr\u00e1nen\u00fd pred svetlom. Po rekon\u0161tit\u00facii v chladni\u010dke pri 2 \u2013 8 \u00b0C, bez opakovan\u00e9ho zmrazovania.<\/p>\n<h3>Kde k\u00fapi\u0165 Tesamorelin na Slovensku?<\/h3>\n<p>V e-shope DoktorPeptid. Tesamorelin peptid 5 mg aj 10 mg m\u00e1me skladom na Slovensku, s COA ku ka\u017edej \u0161ar\u017ei a exped\u00edciou do 24 hod\u00edn. Doru\u010dujeme aj do \u010ceska.<\/p>\n<h3>Je Tesamorelin ur\u010den\u00fd na hum\u00e1nne pou\u017eitie?<\/h3>\n<p>Nie. Produkt je ur\u010den\u00fd v\u00fdhradne na vedeck\u00e9 a laborat\u00f3rne \u00fa\u010dely. Nie je liekom, v\u00fd\u017eivov\u00fdm doplnkom ani potravinou a nie je ur\u010den\u00fd na konzum\u00e1ciu ani na podanie \u013eu\u010fom \u010di zvierat\u00e1m.<\/p>\n<p><strong>Warning:<\/strong> Tesamorelin pred\u00e1vame v\u00fdhradne na v\u00fdskumn\u00e9 a analytick\u00e9 \u00fa\u010dely. Kupuj\u00faci zodpoved\u00e1 za to, \u017ee s l\u00e1tkou bude naklada\u0165 v s\u00falade s platnou legislat\u00edvou a intern\u00fdmi predpismi svojho pracoviska.<\/p>","protected":false},"excerpt":{"rendered":"<p>Tesamorelin skladom na Slovensku. odoslanie do 24 hod\u00edn, doprava SK a \u010cR.<\/p>\n<p><strong>The product is not intended for consumption. For scientific and research purposes only.<\/strong><\/p>","protected":false},"featured_media":668,"comment_status":"closed","ping_status":"closed","template":"","meta":[],"product_brand":[],"product_cat":[33],"product_tag":[],"class_list":["post-432","product","type-product","status-publish","has-post-thumbnail","product_cat-rastove-peptidy","first","instock","taxable","shipping-taxable","purchasable","product-type-variable"],"jetpack_sharing_enabled":true,"_links":{"self":[{"href":"https:\/\/doktorpeptid.sk\/en\/wp-json\/wp\/v2\/product\/432","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/doktorpeptid.sk\/en\/wp-json\/wp\/v2\/product"}],"about":[{"href":"https:\/\/doktorpeptid.sk\/en\/wp-json\/wp\/v2\/types\/product"}],"replies":[{"embeddable":true,"href":"https:\/\/doktorpeptid.sk\/en\/wp-json\/wp\/v2\/comments?post=432"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/doktorpeptid.sk\/en\/wp-json\/wp\/v2\/media\/668"}],"wp:attachment":[{"href":"https:\/\/doktorpeptid.sk\/en\/wp-json\/wp\/v2\/media?parent=432"}],"wp:term":[{"taxonomy":"product_brand","embeddable":true,"href":"https:\/\/doktorpeptid.sk\/en\/wp-json\/wp\/v2\/product_brand?post=432"},{"taxonomy":"product_cat","embeddable":true,"href":"https:\/\/doktorpeptid.sk\/en\/wp-json\/wp\/v2\/product_cat?post=432"},{"taxonomy":"product_tag","embeddable":true,"href":"https:\/\/doktorpeptid.sk\/en\/wp-json\/wp\/v2\/product_tag?post=432"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}